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Volinanserin MDL100907; M 100907

Volinanserin 是一种有效的,选择性的 5-HT2 受体拮抗剂,Ki 值为 0.36 nM,对其选择性是对 5-HT1c,alpha-1 和 DA D2 受体的 300 倍,可用于精神疾病的研究。

  • 货号:
    TK0577
  • 规格:
    1mg
    5mg
    10mg
    25mg
  • 价格:
    0.00

产品参数

CAS No.139290-65-6
生物活性Volinanserin is a potent and selective antagonist of 5-HT2 receptor, with a Ki of 0.36 nM, and shows 300-fold selectivity for 5-HT2 receptor over 5-HT1c, alpha-1 and DA D2 receptors. Volinanserin has antipsychotic activity.
分子式C22H28NO3F
分子量373.46
运输条件Room temperature in continental US; may vary elsewhere.
储存条件Powder -20°C 3 years
溶解性数据DMSO : 50 mg/mL (133.88 mM; Need ultrasonic)