Dapagliflozin 达格列净; BMS-512148
Dapagliflozin (BMS-512148) 是一种竞争性葡萄糖协同转运蛋白2 (SGLT2) 抑制剂,可导致尿液中葡萄糖的排泄,用于糖尿病 (DM) 的研究。Dapagliflozin 诱导 HIF1 表达并减轻肾脏 IR 损伤。
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货号:
TK0575 -
规格:
- 2mg
- 5mg
- 10mg
- 50mg
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价格:
¥0.00
Dapagliflozin (BMS-512148) 是一种竞争性葡萄糖协同转运蛋白2 (SGLT2) 抑制剂,可导致尿液中葡萄糖的排泄,用于糖尿病 (DM) 的研究。Dapagliflozin 诱导 HIF1 表达并减轻肾脏 IR 损伤。
| CAS No. | 461432-26-8 |
| 生物活性 | Dapagliflozin (BMS-512148), a new type of drug used to treat diabetes mellitus (DM), is a competitive sodium/glucose cotransporter 2 (SGLT2) inhibitor, which results in excretion of glucose into the urine. Dapagliflozin induces HIF1 expression and attenuates renal IR injury. |
| 分子式 | C21H25ClO6 |
| 分子量 | 408.87 |
| 运输条件 | Room temperature in continental US; may vary elsewhere. |
| 储存条件 | Powder -20°C 3 years |
| 溶解性数据 | DMSO : ≥ 100 mg/mL (244.58 mM) |